Primodex 50 [10 vials]
General information:
Manufacturer: Sciroxx
Substance: Methenolone Acetate
Pack: 10vials@10ml each (50 mg/ml)
Methenolone Acetate is an anabolic steroid which became very popular
once it was claimed that it was one of Arnold's favorites. I'm not
really sure why this is, or how likely it is that Arnold went around
telling everyone's favorite steroid- but nonetheless, this rumor has
persisted through the years.
When we take a critical look at
it, in terms of its anabolic and androgenic rating, it appears to be a
pretty weak steroid but is rated as stronger than Masteron (
Drostanolone)! I've used
both steroids and can tell you that not too many people would claim
that those ratings provide an accurate idea of those two steroids
compare to each other. In truth, I used Primobolan at 400mgs/week and
wasn't very impressed with it, and honestly, for the money, that's
really disappointing, since
Primobolan is not
inexpensive. I also would speculate that the reason many (male)
Primobolan users have been less than thrilled with results from it is
that they failed to use high enough doses. If I were to use it again
(which I won't), I would probably use 100mgs/ED (Every Day).
Interestingly,
Primobolan
has a relatively high affinity for binding to the Androgen Receptor,
and surprisingly it actually binds with more affinity than testosterone
(1). This ability to strongly bind to the AR may be why Primobolan is
considered a good fat burner- although most Dihydrotestosterone (DHT)
derivations are very potent fat burners (the notable exception being
Anadrol).
Primobolan has been used medically to reduce breast
tumors, with a success rate of about a third (2), so we can safely
assume that no Anti-Estrogen products would be necessary. The use of
Finasteride, Dutesteride, or another anti-hair-loss product may be useful, however, as
Primobolan has a bad reputation for causing Alopecia.
Primobolan is very useful as both an anabolic as well as anti-catabolic
agent, and the probable cause for this property is its ability to aid
in nitrogen retention (3), which is a useful trait on both a bulking or
cutting cycle?once again, I have to reiterate that the expense of this
drug probably makes it a poor choice on a bulking cycle because of the
reasonably high doses that it would require.
One of the other very interesting facts about Primobolan is that it's
one of the very few compounds available as both an oral as well as an
injectable. Unlike Winstrol and Dianabol (both alkylated and
non-estrified steroids) however, which are also available in both
forms, Primobolan is available with an Acetate ester for use as an
oral, and with an Enanthate ester as an injectable. Unfortunately, in
this case, making Primobolan a non-17-alpha-alkylated steroid greatly
reduces its potency. However, it must be noted that this alkylation is
what makes oral steroids survive their first pass through the liver; it
also makes them hepatoxic (liver toxic). Oral Primobolan doesn't
actually have this drawback, and thus it is very mild on liver function
and doesn't elevate liver enzymes too much. Instead of the more toxic
17a-alkylation, Primobolan (Oral) uses 17 beta estrification and 1
alkylation to make it orally available. For both men as well as women,
daily dosing of the oral is necessary, although men would probably want
to take 100mgs per day and women would need to take at least 10mgs
every day.
Although it is typically considered to be a very mild drug when
inhibition of the natural hormonal profile is considered, this isn't
totally true. Men were given a 30-45mg dose of the oral version of
Primobolan, experienced between a 15% and 65% decrease in their
Gonadatropin levels (4). Since we're probably looking at double or
triple that dose, for men to get any kind of results, it?s also
probable that gonadal inhibition will also be increased.
My history with Primobolan Enanthate (the injectable version) has been
less than impressive. I used it at 200mgs/week about a decade ago, and
wasn't impressed at all. A couple of years ago I went back to it and
used 350mgs/week (100mgs/Every other Day), and got much better results,
but still wasn't overly impressed with it. Add to that the fact that it
is an expensive chemical, and I really wasn't impressed.
On the Black Market, Primobolan tabs are only being produced by
British Dragon
currently, although PaperPrimo is being produced as well. Both are high
quality products, although I would speculate that their use is going to
be reserved for women. With regards to the injectable version, many
underground labs produce it, and quality tends to vary, due to powder
quality at the moment. Expect to pay around $100 for a 10ml bottle
dosed at 100mgs/ml, if not more. Finally, ampules are available at a
cost of roughly $7-12 per amp, but since this is the most widely
counterfeited steroid on the black market, I'd stick to the underground lab variety.
References:
1.
Relative binding affinity of anabolic-androgenic steroids: comparison
of the binding to the androgen receptors in skeletal muscle and in
prostate, as well as to sex hormone-binding globulin. Endocrinology.
1984 Jun;114(6):2100-6.
2.
Med Klin. 1981 Nov 20;76(24):689-91. [Anabolic therapy in metastatic
breast cancer] [Article in German] Hartmann F, Pompecki R, Desaga U,
Frahm H
3.
Metabolic effects of anabolic steroids. Wien Med Wochenschr.
1993;143(14-15):368-75 Anabolic steroids (metenolone) improve muscle
performance and hemodynamic characteristics in cardiomyoplasty.
4.
Comparative Studies about the influence of MetenoloneAcetate and
Mesterolone on hypophysis and male gonads. Arzneimittelforshung. 1970
20(4) 545-7 Ann Thorac Surg. 1995 Apr;59(4):961-9; discussion 969-70.